Important Safety Information

Microdose GLP-1 — Important Safety Information

Low-dose GLP-1 therapy. Same class warnings apply as compounded semaglutide and tirzepatide.

Last reviewed:

Compounded drugs are permitted to be prescribed under federal law, but are not FDA-approved and do not undergo FDA safety, effectiveness, or manufacturing review. Your EOS Health-affiliated provider may recommend this medication based on your individual medical evaluation.

Microdose GLP-1 may use either compounded semaglutide or compounded tirzepatide depending on your individual treatment plan. The same class warnings apply as the full-dose versions of these medications. Please review the section that applies to your prescribed treatment, and consult your EOS Health-affiliated provider with any questions.

Important Safety Information for Compounded Tirzepatide

Contraindications

Tirzepatide is contraindicated in patients with a personal or family history of medullary thyroid carcinoma (MTC) or Multiple Endocrine Neoplasia syndrome type 2 (MEN 2). It should not be used in patients with a history of severe gastrointestinal disease, including gastroparesis.

Warnings and Precautions

  1. Risk of Thyroid C-Cell Tumors: Cases of MTC have been reported with GLP-1 receptor agonists.
  2. Pancreatitis: Acute pancreatitis has been reported. Discontinue and seek medical attention if symptoms occur.
  3. Hypoglycemia when used with insulin or insulin secretagogues.
  4. Acute Kidney Injury: Monitor renal function.
  5. Hypersensitivity Reactions including anaphylaxis, angioedema, urticaria.
  6. Gastrointestinal Adverse Reactions: Nausea, vomiting, diarrhea, constipation.

Most common reactions: nausea, vomiting, diarrhea, abdominal pain, constipation.

Pregnancy: Should not be used. Caution in breastfeeding.


Important Safety Information for Compounded Semaglutide

Warning: Risk of Thyroid C-Cell Tumors

  • Semaglutide caused thyroid tumors in mice and rats. Tell your provider about any neck lump or swelling, hoarseness, trouble swallowing, or shortness of breath.
  • Do not use if you or family have ever had MTC or MEN 2.

Who should not use semaglutide?

  • Personal or family history of MTC or MEN 2
  • Known allergic reaction to semaglutide

What to tell your provider

Share all medications and your full medical history, especially: diabetes, thyroid cancer, pancreatitis, kidney disease, diabetic retinopathy, depression, suicidal thoughts.

Most serious side effects

If experiencing a medical emergency, call 911.

  • Thyroid C-cell tumors
  • Acute pancreatitis
  • Acute gallbladder disease
  • Low blood sugar (hypoglycemia)
  • Acute kidney injury
  • Serious allergic reactions
  • Diabetic retinopathy complications
  • Increased heart rate
  • Suicidal behavior and ideation
  • Never share needles or syringes

Most common side effects

  • Nausea, diarrhea, vomiting, constipation, abdominal pain, headache, fatigue, dyspepsia, dizziness.

Pregnancy and breastfeeding

  • Should not be used during pregnancy.
  • Discontinue at least 2 months before a planned pregnancy.

You are encouraged to report negative side effects to FDA MedWatch: www.fda.gov/medwatch or 1-800-FDA-1088.

This information is not comprehensive. Please reach out to your EOS Health-affiliated provider with any questions or concerns.